 COA |
MSDS |
 HPLC |
NMR |
| CAS No: | 1620401-82-2 |
| Molecular formula(MF) | C23H35N5O2 |
| Molecular Weight(MW): | 413.56 |
| Alias |
| Description | UNC0379 is a selective, substrate competitive inhibitor of N-lysine methyltransferase SETD8 with IC50 of 7.9 μM, high selectivity over 15 other methyltransferases. | ||
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| Targets |
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| In vitro |
UNC0379 is competitive with the peptide substrate and noncompetitive with the cofactor SAM. [1] |