GSK1278863
(CAS No:960539-70-2)
QC Documents
ChemicalInfomation
CAS No: |
960539-70-2 |
Molecular formula(MF) |
C19H27N3O6 |
Molecular Weight(MW): |
393.43 |
Alias |
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Solubility
In vitro |
DMSO
|
10 mg/mL
warmed
(25.41 mM)
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Water
|
<1 mg/mL
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Ethanol
|
<1 mg/mL
|
In vivo |
|
|
Biological Activity
Description |
Daprodustat (GSK1278863) is an orally administered hypoxia-inducible factor-prolyl hydroxylase (HIF-PH) inhibitor. Phase 2.
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Targets
|
|
In vitro |
GSK1278863 induces an effective EPO response and stimulates non-EPO mechanisms for erythropoiesis. [1]
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